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Contents





                    Preface  vii
                    Authors  ix



                    S ECTI O N  I                                        10.  Adrenoceptor Antagonist Drugs
                                                                             David Robertson, MD, & Italo Biaggioni, MD  156
                    BASIC PRINCIPLES    1                                S ECTI O N  III


                      1.  Introduction: The Nature of Drugs &            CARDIOVASCULAR-RENAL
                        Drug Development & Regulation
                        Bertram G. Katzung, MD, PhD  1                   DRUGS   173

                      2.  Drug Receptors & Pharmacodynamics              11.  Antihypertensive Agents
                        Mark von Zastrow, MD, PhD  20                        Neal L. Benowitz, MD  173

                      3.  Pharmacokinetics & Pharmacodynamics:           12.  Vasodilators & the Treatment of
                        Rational Dosing & the Time Course                    Angina Pectoris
                        of Drug Action                                       Bertram G. Katzung, MD, PhD  194
                        Nicholas H. G. Holford, MB, ChB, FRACP  41
                                                                         13.  Drugs Used in Heart Failure
                      4.  Drug Biotransformation                             Bertram G. Katzung, MD, PhD  212
                        Maria Almira Correia, PhD  56
                                                                         14.  Agents Used in Cardiac Arrhythmias
                      5.  Pharmacogenomics                                   Robert D. Harvey, PhD,
                        Jennifer E. Hibma, PharmD,                           & Augustus O. Grant, MD, PhD  228
                        & Kathleen M. Giacomini, PhD  74
                                                                         15.  Diuretic Agents
                    S ECTI O N  II                                           Ramin Sam, MD, Harlan E. Ives, MD, PhD,
                                                                             & David Pearce, MD  254

                    AUTONOMIC DRUGS    89                                S ECTI O N  IV

                      6.  Introduction to Autonomic Pharmacology         DRUGS WITH IMPORTANT ACTIONS
                        Bertram G. Katzung, MD, PhD  89
                                                                         ON SMOOTH MUSCLE    277
                      7.  Cholinoceptor-Activating &
                        Cholinesterase-Inhibiting Drugs                  16.  Histamine, Serotonin, & the Ergot Alkaloids
                        Achilles J. Pappano, PhD   107                       Bertram G. Katzung, MD, PhD  277

                      8.  Cholinoceptor-Blocking Drugs                   17.  Vasoactive Peptides
                        Achilles J. Pappano, PhD  124                        Ian A. Reid, PhD  300

                      9.  Adrenoceptor Agonists &                        18.  The Eicosanoids: Prostaglandins,
                        Sympathomimetic Drugs                                Thromboxanes, Leukotrienes, & Related
                        Italo Biaggioni, MD, & David Robertson, MD  137      Compounds
                                                                             John Hwa, MD, PhD, &
                                                                             Kathleen Martin, PhD  321


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