Page 950 - Basic _ Clinical Pharmacology ( PDFDrive )
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936     SECTION VIII  Chemotherapeutic Drugs


                 PREP AR A TIONS                                     German PI, Aweeka FT: Clinical pharmacology of artemisinin-based combination
                                                                         therapies. Clin Pharmacokinet 2008;47:91.
                 A V AIL ABLE                                        Hill DR et al: Primaquine: Report from CDC expert meeting on malaria chemo-
                                                                         prophylaxis I. Am J Trop Med Hyg 2006;75:402.
                      GENERIC NAME             AVAILABLE AS          John GK et al: Primaquine radical cure of Plasmodium vivax: A critical review of
                                                                         the literature. Malar J 2012;11:280.
                 Artemether/lumefantrine  Coartem, Riamet            McGready R et al: Adverse effects of falciparum and vivax malaria and the safety of
                 Artesunate *                                            antimalarial treatment in early pregnancy: A population-based study. Lancet
                 Artesunate-pyronaridine  Pyramax                        Infect Dis 2012;12:388.
                 Atovaquone            Generic, Mepron               Morris CA et al: Review of the clinical pharmacokinetics of artesunate and its
                                                                         active metabolite dihydroartemisinin following intravenous, intramuscular,
                 Atovaquone-proguanil  Malarone                          oral or rectal administration. Malar J 2011;10:263.
                 Benznidazole *                                      Nadjm B, Behrens RH: Malaria: An update for physicians. Infect Dis Clin North
                 Chloroquine           Generic, Aralen                   Am 2012;26:243.
                 Clindamycin           Generic, Cleocin              Nosten F et al: Antimalarial drugs in pregnancy: A review. Curr Drug Saf 2006;1:1.
                 Doxycycline           Generic, Vibramycin           Rehman K, et al: Haemolysis associated with the treatment of malaria with arte-
                                                                         misinin derivatives: a systematic review of current evidence. Int J Infect Dis
                 Eflornithine          Vaniqa, Ornidyl                   2014;29:268.
                 Iodoquinol            Diquinol, Yodoxin             Rosenthal PJ: Artesunate for the treatment of severe falciparum malaria. N Engl J
                 Mefloquine            Generic, Lariam                   Med 2008;358:1829.
                 Melarsoprol *         Mel B                         Rosenthal PJ: The interplay between drug resistance and fitness in malaria para-
                                                                         sites. Mol Microbiol 2013;89:1025.
                 Metronidazole         Generic, Flagyl               Stepniewska K,  White NJ: Pharmacokinetic determinants of the window of
                 Nifurtimox *                                            selection for antimalarial drug resistance. Antimicrob Agents Chemother
                 Nitazoxanide          Alinia                            2008;52:1589.
                 Paromomycin           Generic, Humatin              Taylor WR, White NJ: Antimalarial drug toxicity: A review. Drug Saf 2004;
                 Pentamidine           Pentam 300, Pentacarinat, pentami-  27:25.
                                       dine isethionate, Nebupent (aerosol)  Tilley L et al: Artemisinin Action and Resistance in Plasmodium falciparum. Trends
                                                                         Parasitol 2016 32:682.
                 Primaquine            Generic                       White NJ: Cardiotoxicity of antimalarial drugs. Lancet Infect Dis 2007;7:549.
                 Pyrimethamine         Daraprim                      White NJ et al: Malaria. Lancet 2014;383:723.
                 Quinidine gluconate   Generic                       Whitty CJ, Chiodini PL, Lalloo DG: Investigation and treatment of imported
                 Quinine               Generic                           malaria in non-endemic countries. BMJ 2013;346:f2900.
                 Sodium stibogluconate *                             World Health Organization: Guidelines for the treatment of malaria. Geneva.
                 Sulfadoxine-pyrimethamine  Fansidar                     2015. www.who.int/malaria/publications/atoz/9789241549127/en/.
                 Suramin *              
                 Tinidazole            Generic, Tindamax             Intestinal Protozoal Infections
                                                                     Fox LM, Saravolatz LD: Nitazoxanide: A new thiazolide antiparasitic agent. Clin
                 * Available in the USA only from the Drug Service, CDC, Atlanta, Georgia (phone:   Infect Dis 2005;40:1173.
                 404-639-3670; www.cdc.gov/laboratory/drugservice/).
                                                                     Granados CE et al: Drugs for treating giardiasis. Cochrane Database Syst Rev
                                                                         2012;(12):CD007787.
                 REFERENCES                                          Leitsch D: Drug resistance in the microaerophilic parasite Giardia lamblia. Curr
                                                                         Trop Med Rep 2015;2:128.
                 General                                             Marcos LA, Gotuzzo E: Intestinal protozoan infections in the immunocompro-
                                                                         mised host. Curr Opin Infect Dis 2013;26:295.
                 Kappagoda S, Singh U, Blackburn BG: Antiparasitic therapy. Mayo Clin Proc   Pierce KK et al: Update on human infections caused by intestinal protozoa. Curr
                    2011;86:561.                                         Opin Gastroenterol 2009;25:12.
                 Medical Letter: Drugs for parasitic infections. Med Lett Drugs  Ther   Pritt BS, Clark DG: Amebiasis. Mayo Clin Proc 2008;83:1154.
                    2013;Supplement.
                                                                     Ross AG et al: Enteropathogens and chronic illness in returning travelers. N Engl
                                                                         J Med 2013;368:1817.
                 Malaria                                             Rossignol JF: Cryptosporidium and Giardia: Treatment options and prospects for
                 Ashley EA et al: Tracking Resistance to Artemisinin Collaboration (TRAC). Spread   new drugs. Exp Parasitol 2010;124:45.
                    of artemisinin resistance in Plasmodium falciparum malaria. N Engl J Med   Wright SG: Protozoan infections of the gastrointestinal tract. Infect Dis Clin
                    2014;371:411.                                        North Am 2012;26:323.
                 Baird KJ, Maguire JD, Price RN: Diagnosis and treatment of Plasmodium vivax
                    malaria. Adv Parasitol 2012;80:203.              Trypanosomiasis & Leishmaniasis
                 Boggild AK et al: Atovaquone-proguanil: Report from the CDC expert meeting on
                    malaria chemoprophylaxis (II). Am J Trop Med Hyg 2007;76:208.  Aronson NE et al: A randomized controlled trial of local heat therapy versus intra-
                 Bukirwa H et al: Artesunate plus pyronaridine for treating uncomplicated Plasmo-  venous sodium stibogluconate for the treatment of cutaneous Leishmania
                    dium falciparum malaria. Cochrane Database Syst Rev 2014;(3):CD006404.  major infection. PLoS Negl Trop Dis 2010;4:e628.
                 Dondorp AM et al: Artesunate versus quinine in the treatment of severe falciparum   Ben Salah A et al: Topical paromomycin with or without gentamicin for cutaneous
                    malaria in African children (AQUAMAT): An open-label, randomised trial.   leishmaniasis. N Engl J Med 2013;368:524.
                    Lancet 2010;376:1647.                            Bern C: Chagas’ disease. N Engl J Med 2015;373:456.
                 Efferth T, Kaina B: Toxicity of the antimalarial artemisinin and its derivatives. Crit   Bhattacharya SK et al: Phase 4 trial of miltefosine for the treatment of Indian
                    Rev Toxicol 2010;40:405.                             visceral leishmaniasis. J Infect Dis 2007;196:591.
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