Page 143 - MNU-PM502- Pharmaeutical Microbiology Theoritical Book
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Pharm D- Clinical Pharmacy Program        Third Level          Pharmaceutical Microbiology& Antimicrobials (PM 502)


                   Nucleoside  Reverse  Transcriptase  Non-Nucleoside Reverse
                   Inhibitor                                     Transcriptase Inhibitor

                   competitive  inhibitors  of  reverse  Non-competitive  inhibitors  of  reverse
                   transcriptase.                                transcriptase
                       ➢  Zidovudine                                 ➢  Nevirapine

                       ➢  Stavudine                                  ➢  Efavirenz
                       ➢  Lamivudine
                       ➢  Tenofovir

                       3. Integrase inhibitor
                   Interfere with integrase enzyme which inserts HIV genetic material into human
                   cell.

                       ➢  Raltegravir


                       4. Protease Inhibitors
                       ➢  Indinavir                     ➢  Atazanavir,  darunavir,  lopinavir,
                       ➢  Saquinavir
                                                            nelfinavir, ritonavir



































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