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328              MEDICAMENTINDUISANT OUSTABILISANTDES COUPURES DE L'ADN


             MINISCI F. et PORTA O., Advances in Heterocyclic Chem., 1974, 16, 1713-1718.
             WANI M. et al., Synthesis and biological activity of camptothecin analogues, J. Med.
               Chem., 1980, 23, 554-560.
             WANI M. et al., Isolation of 11-hydroxycamptothecin from Camptotheca acuminata, total
               synthesis and biological activity, J. Med. Chem., 1986, 29, 1553-1555.
             KINGSBURY W., Synthesis of water-soluble (aminoalkyl)camptothecin analogues,J. Med.
               Chem., 1991, 34, 98-107.
             SAWADA S. et al., Synthesis and antitumor activity of 20(S)-camptothecin derivatives,
               Chem. Pharm. Bull., 1991, 39, 1446-1454.
             SAWADA S. et al., Synthesis and antitumor activity of 7-C-substituted camptothecins,
             Chem. Pharm. Bull., 1991, 39, 2574-2580.

             IRINOTÉCAN
              YAKULT HONSHA Co, brevets Jap. 85 19.790 (1985) et US 4.604.463.
              KAWATO Y. et al., Intracellular roles of SN-38, a metabolite of the camptothecin derivate
               CPT-11, CancerRes., 1991, 51, 4187-4191.
              KAWATO Y. et al., Antitumor activity of CPT-11, against human tumor xenografts in nude
               mice, Cancer Chemother. Pharmacol., 1991, 28, 192-198.
              SAWADA S. et al., A-ring modified and 7,10-disubstituted camptothecins, Chem. Pharm.
               Bull., 1991, 39, 3183-3188.
              RIVORY L et ROBERT J., Molecular, cellular and clinical aspects of the pharmacology
                of camptothecin and its derivatives, Pharmacol. Ther., 1995, 68, 269-296 ; Pharma-
                cologie de la camptothécine et de ses dérivés, Bull. Cancer, 1995, 82, 265-285 ; Iden-
                tification and kinetics of a glucuronide metabolite of SN-38 in human plasma after
                administration of the camptothecin derivate irinotecan, Cancer Chemother. Pharma-
                col., 1995, 36, 176-179.
              SAWADA S. et al., Synthesis of CPT-11, Ann. N.Y. Acad. Sci., 1996, 803, 13-28.
              Society of Japanese Pharmacopoiea/Japanese Ministry of Health and Welfare, Summary
                Basis of approval for lrinotecan hydrochloride, YAKUJI NIPPO Ltd, Tokyo, 1996.
              BEDESCHI A. et al., Water-soluble camptothecin derivatives, Drugs Future, 1997, 22,
                1259-1266.
              TOPOTÉCAN
              SMITHKLINE Co, brevet européen 321.122 (1989).
              CABRI W. et al., New high yield semisynthetic approach to 9-aminocamptothecin, Tetra-
                hedron Lett., 1995, 36, 9197-9200.
              CREEMERS G. et al., Topotecan, an active drug in the second-line treatment of epithelial
                ovarian cancer, J. Clin. Oncol., 1996, 14, 3056-3061.
               HERBEN V. et al., Clinlcal pharmacokinetlcs of topotecan, Clin. Pharmacokinetic., 1996,
                31, 85-102.
               European Agency for the Evaluation of Medicinal Products, rapports EPAR-CPMP
                709/96 et 642/96, Londres, 1996.
               KUDELKA A. et al., Phase Il study of lntravenous topotecan, J. Clln. Oncol., 1996, 14,
                1552-1557.
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