Page 450 - Traité de chimie thérapeutique 6 Médicaments antitumoraux
P. 450
406 MEDICAMENTS INDUISANTOUSTABILISANTDES COUPURES DE L'ADN
ARCAMONE F. et al., Daunomycin Il. The structure and stereochemistry of daunosamine,
J. Am. Chem. Soc., 1964, 86, 5335-5336.
IWAMOTO R. H. et al., The structure of daunomycin, Tetrahedron Letters, 1968, 36,
3891-3894.
ARCAMONE F. et al., Struttura e stereochimica della daunomicina, Gazz. Chim. /ta/.,
1970, 100, 949-989.
WONG C.M. et al., Synthetic studies of hydronaphthacenic antibiotics 1. The synthesis
of 4-demethoxy-7-O-methyldaunomycinone, Can. J. Chem., 1971, 49, 2712-2718.
ACTON E. M. et al., Total synthesis of the antitumor antibiotic daunorucicin. Coupling of
the sugar and aglycone. J. Med. Chem., 1974, 17, 659-660.
ARCAMONE F. et al., Synthesis and antitumor properties of new glycosides of dauno-
mycinone and adriamycinone, J. Med. Chem., 1975, 18, 703-707.
ARCAMONE F. et al., Synthesis and antitumor activity of 4-demethoxydaunorubicin, 4-
demethoxy-7,9-diepidaunorubicin, and theiranomers, CancerTreat. Rep., 1976, 60,
829-834.
SUZUKI F. et al., Total synthesis of adriamycinone. Regiospecific synthesis of anthracy-
clinones via base-catalyzed cyclizations, J. Am. Chem. Soc., 1978, 100, 2272-2273.
SWENTON J.S., RAYNOLDS P.W., A regiospecific synthesis of the anthracycline aglyco-
nes, daunomycinone and adriamycinone, J. Am. Chem. Soc., 1978, 100, 6188-6195.
UMEZAWA H. et al., Tetrahydropyranyl derivatives of daunomycin and adriamycin, J.
Antibiotics, 1979, 32, 1082-1084.
ARDECKY R. J. et al., 3-(Acyloxy)-3-buten-2-ones as dienophiles in anthracyclinone syn-
thesis. An efficient route to 4-demethoxy-7-deoxydaunomycinone derivatives, J. Org.
Chem., 1982, 47, 409-412.
BROADHURST M. J., HASSAL C. H., Anthracyclines. The synthesis of racemic dauno-
mycinone and some related tetrahydronaphtacenequinones, J. Chem. Soc., Perkin
Trans 1, 1982, 2227-2238.
BROADHURST M. J. et al., Anthracyclines. Investigations relating to the synthesis of 4-
demethoxyanthracyclinones, J. Chem. Soc. Perkin Trans. 1, 1982, 2239-2248.
BROADHURST M. J. et al., Anthracyclines. The total synthesis of 4-demethoxydauno-
mycin, J. Chem. Soc. Perkin Trans. 1, 1982, 2249-2255.
GRETHE G. et al., Synthesis of daunosamine, J. Org. Chem., 1983, 48, 5309-5315.
GRETHE G. et al., Asymmetric synthesis of daunosamine, J. Org. Chem., 1983, 48,
5315-5317.
BROADHURST M. J. et al., Total synthesis of some new 4-demethoxyanthracyclinones,
Tetrahedron, 1984, 22, 4656-4649.
CARDILLO G. et al., Regio- and stereoselective synthesis of methyl a-L-daunosaminide
hydrochloride, J. Org. Chem., 1984, 49, 3951-3953.
DESHONG P. et al., Stereoselection in acyclic systems. The synthesis of amino sugars
via nitrone cycloadditions, J. Am. Chem. Soc., 1984, 106, 5598-5602.
UMEZAWA H. et al., The absolute structures of THP-adriamycins, J. Antibiotics, 1984,
37, 1094-1097.
WOVKULICH P.M., USKOKOVIC M.R., Total synthesis of acosamine and daunosamine
utilizing a diastereoselective intramolecular (3+2] cycloaddation, Tetrahedron, 1985,
17, 3455-3462.